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Our mission is to change this by creating the most trusted place to discover curated, quality-assessed health & wellness products from around the world.

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How our curation process works

2

Evaluate

Each product then undergoes a comprehensive vetting process over a six-week period. This extensive time window allows us to delve into the details of each standard. Brands are ultimately signed off on by our review committee of leading doctors, scientists, and pharmacologists.

We evaluate products across 11 factors, here are a few of our most important:

2.1 Evaluate

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500+

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View our list of sources

These sources are valuable for evaluating the safety and non-toxicity of products, providing consumers with reliable information to make informed choices.

Environmental Working Group (EWG)

EWG is known for providing tools and resources to make better choices regarding toxic-free, safe products in various categories, including household and consumer products.

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ConsumerLab is known for its comprehensive set of test results, including dosage, phytonutrient levels, and contaminant levels in various products.

Examine

ConsumerLab is known for its comprehensive set of test results, including dosage, phytonutrient levels, and contaminant levels in various products.

NSF Supplement Vitamin Certification

ConsumerLab is known for its comprehensive set of test results, including dosage, phytonutrient levels, and contaminant levels in various products.

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ConsumerLab is known for its comprehensive set of test results, including dosage, phytonutrient levels, and contaminant levels in various products.

Lab Door

ConsumerLab is known for its comprehensive set of test results, including dosage, phytonutrient levels, and contaminant levels in various products.
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3

Monitor

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Oxytocin/ Bremelanotide/ Tadalafil
RX

Oxytocin/ Bremelanotide/ Tadalafil

Rediscover your passion with a powerful blend designed to enhance intimacy, boost libido, and elevate your confidence.

Personalized Prescription

Free Priority Shipping

Ongoing Care & Support

Oxytocin/ Bremelanotide/ Tadalafil
Oxytocin/ Bremelanotide/ Tadalafil Default Title

The science of Oxytocin/ Bremelanotide/ Tadalafil

Active ingredients


* Oxytocin (40 IU)* Bremelanotide (2 mg)* Tadalafil (20 mg)

Mechanism


Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

History


Tadalafil was approved by the FDA in 2003 for erectile dysfunction and later for benign prostatic hyperplasia (BPH). Compounding pharmacies have more recently started formulating troches combining these agents to address sexual function in a more holistic manner.

Frequently Asked Questions

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

Am I a good candidate?

You may be a candidate if you:

  • Struggle with low libido (in men or women).
  • Experience difficulty achieving or maintaining erections (in men).
  • Want to address multiple aspects of sexual function (desire, arousal, vascular support).
  • Have discussed potential options with a licensed healthcare provider and have no contraindications.
  • You may not be a good candidate if you: Have underlying medical conditions (e.g., significant heart issues, low blood pressure, uncontrolled hypertension, or severe liver/kidney disease) without proper medical oversight.
  • Are taking certain medications (e.g., nitrates) that could dangerously interact with tadalafil.
  • Are pregnant, nursing, or planning to become pregnant—safety data are not well-established for these populations.

What states is this available in?

CA, FL, NY, TX, CO, NV, NJ

Supporting science and sources

Oxytocin research shows it can modulate social and sexual behaviors by acting on brain receptors that influence bonding and arousal.



Bremelanotide studies demonstrate an increase in sexual desire and satisfaction in some individuals, particularly for hypoactive sexual desire disorder.



Tadalafil and other PDE5 inhibitors have a well-documented history of treating erectile dysfunction through enhanced nitric oxide-mediated vasodilation.

How do I use Oxytocin/ Bremelanotide/ Tadalafil?

Troches (lozenges) are placed under the tongue or in the cheek (buccal area) and allowed to dissolve.

Timing:

  • Tadalafil is often taken at least 30 minutes to 1 hour before sexual activity for optimal effect.
  • Bremelanotide/oxytocin may have varying onset times. Take 90-120 minutes prior to sexual activity

How does Oxytocin/ Bremelanotide/ Tadalafil effect my body?

  • Absorption: When taken as a troche, the medication is absorbed through the oral mucosa, bypassing part of the gastrointestinal tract and first-pass metabolism.
  • Distribution: Tadalafil is distributed systemically to improve blood flow, while bremelanotide primarily exerts its effect in the central nervous system and peripheral melanocortin receptors. Oxytocin also has central and peripheral mechanisms of action but is typically short-acting.
  • Metabolism: Tadalafil is metabolized in the liver (primarily by CYP3A4). Bremelanotide and oxytocin are broken down by enzymes in the bloodstream and various tissues.
  • Elimination: Tadalafil’s half-life is around 17.5 hours, whereas oxytocin and bremelanotide have shorter half-lives and are excreted primarily via the kidneys.

Special Considerations

  • Blood Pressure: Tadalafil can cause a mild drop in blood pressure. Use caution if you have cardiovascular conditions or if you are taking medications that affect blood pressure.
  • Allergies: Alert your healthcare provider if you have known allergies to any component (e.g., dyes or flavors in the troche).
  • Medical Conditions: Discuss all medical conditions with your healthcare provider, especially heart disease, liver or kidney impairment, uncontrolled hypertension, and prior or existing strokes or heart attacks.
  • Pregnancy and Nursing: Safety for pregnant or breastfeeding individuals is not established.

How do I safely store Oxytocin/ Bremelanotide/ Tadalafil?

Store the troches in a cool, dry place away from direct light and heat. Keep out of reach of children and pets. Follow any specific storage instructions provided by the compounding pharmacy (e.g., refrigeration if recommended).

What if I miss a dose?

Since this is typically used “as needed,” missing a scheduled dose is less common. However, follow your healthcare provider’s instructions. Do not double dose to make up for a missed dose. Take only as prescribed.

Can women use this troche?

Yes, in certain cases. Bremelanotide and oxytocin are studied for female sexual response, and while tadalafil is primarily indicated for erectile dysfunction in men, there is ongoing research exploring its effects on blood flow and sexual arousal in women. Consult a healthcare professional to determine if this therapy is appropriate for you.

How quickly will I feel the effects?

Response time can vary among individuals. Tadalafil often begins working within 30–60 minutes, while bremelanotide/oxytocin effects on libido may be more gradual and variable. Your prescribing provider can give more personalized information based on your health profile.

What does off-label usage mean?

Off-label usage refers to the practice of prescribing or using a medication, medical device, or treatment for a purpose that is not approved by regulatory authorities, such as the FDA (Food and Drug Administration) in the United States. This means that the medication is being used in a manner or for a condition that is not specifically listed on its label or approved product information. Off-label usage may occur when healthcare professionals believe that the treatment may be beneficial for a particular condition, based on clinical judgment, research, or anecdotal evidence, even if it has not been formally approved for that specific use.

For Superpower Members, text your private concierge at any time with any question

Important safety information

Potential Side Effects

Potential side effects can include:

  • Headache
  • Flushing
  • Nausea (sometimes associated with bremelanotide)
  • Nasal congestion
  • Upset stomach or reflux
  • Dizziness or lightheadedness
  • Skin changes (rare, but possible with melanocortin agonists like bremelanotide)
  • Most side effects are mild and transient. If you experience severe or persistent side effects (e.g., severe drop in blood pressure, irregular heartbeat, prolonged erections), seek medical attention promptly.

Contraindications

  • Concurrent use of nitrates (e.g., nitroglycerin) can lead to dangerously low blood pressure.
  • Severe liver or kidney impairment without close medical supervision.

    Uncontrolled hypertension or hypotension.
  • History of serious cardiac events (e.g., recent stroke or myocardial infarction) without clearance from a cardiologist.
  • Allergic reactions: If you have a known hypersensitivity to any component (oxytocin, bremelanotide, tadalafil, or excipients), avoid use.

Drug Interactions

  • Nitrates (e.g., nitroglycerin) or alpha-blockers can cause significant blood pressure drops when combined with tadalafil.
  • Certain CYP3A4 inhibitors (e.g., some antibiotics, antifungals) can increase the concentration of tadalafil.
  • Alcohol: Excessive alcohol may amplify certain side effects like dizziness and hypotension.

Potential Side Effects

Potential side effects can include:

  • Headache
  • Flushing
  • Nausea (sometimes associated with bremelanotide)
  • Nasal congestion
  • Upset stomach or reflux
  • Dizziness or lightheadedness
  • Skin changes (rare, but possible with melanocortin agonists like bremelanotide)
  • Most side effects are mild and transient. If you experience severe or persistent side effects (e.g., severe drop in blood pressure, irregular heartbeat, prolonged erections), seek medical attention promptly.

Contraindications

  • Concurrent use of nitrates (e.g., nitroglycerin) can lead to dangerously low blood pressure.
  • Severe liver or kidney impairment without close medical supervision.

    Uncontrolled hypertension or hypotension.
  • History of serious cardiac events (e.g., recent stroke or myocardial infarction) without clearance from a cardiologist.
  • Allergic reactions: If you have a known hypersensitivity to any component (oxytocin, bremelanotide, tadalafil, or excipients), avoid use.

Drug Interactions

  • Nitrates (e.g., nitroglycerin) or alpha-blockers can cause significant blood pressure drops when combined with tadalafil.
  • Certain CYP3A4 inhibitors (e.g., some antibiotics, antifungals) can increase the concentration of tadalafil.
  • Alcohol: Excessive alcohol may amplify certain side effects like dizziness and hypotension.

Potential Side Effects

Potential side effects can include:

  • Headache
  • Flushing
  • Nausea (sometimes associated with bremelanotide)
  • Nasal congestion
  • Upset stomach or reflux
  • Dizziness or lightheadedness
  • Skin changes (rare, but possible with melanocortin agonists like bremelanotide)
  • Most side effects are mild and transient. If you experience severe or persistent side effects (e.g., severe drop in blood pressure, irregular heartbeat, prolonged erections), seek medical attention promptly.

Contraindications

  • Concurrent use of nitrates (e.g., nitroglycerin) can lead to dangerously low blood pressure.
  • Severe liver or kidney impairment without close medical supervision.

    Uncontrolled hypertension or hypotension.
  • History of serious cardiac events (e.g., recent stroke or myocardial infarction) without clearance from a cardiologist.
  • Allergic reactions: If you have a known hypersensitivity to any component (oxytocin, bremelanotide, tadalafil, or excipients), avoid use.

Drug Interactions

  • Nitrates (e.g., nitroglycerin) or alpha-blockers can cause significant blood pressure drops when combined with tadalafil.
  • Certain CYP3A4 inhibitors (e.g., some antibiotics, antifungals) can increase the concentration of tadalafil.
  • Alcohol: Excessive alcohol may amplify certain side effects like dizziness and hypotension.

For Superpower Members, text your private concierge at any time with any question

Our Curation Standards

At Superpower, we believe in scientific rigor and transparency. We have a dedicated medical and research team that follows a multi-faceted curation and evaluation process to select only the most trusted and efficacious products and protocols for our members.

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